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Assay Detail

CHEMBL5029450

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity to human CREBBP bromodomain expressed in Escherichia coli BL21 (DE3)-RIL
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

CREB-binding protein (CHEMBL5747)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Controlling Intramolecular Interactions in the Design of Selective, High-Affinity Ligands for the CREBBP Bromodomain.
Brand M, Clayton J, Moroglu M, Schiedel M, Picaud S, Bluck JP, Skwarska A, Bolland H, Chan AKN, Laurin CMC, Scorah AR, See L, Rooney TPC, Andrews KH, Fedorov O, Perell G, Kalra P, Vinh KB, Cortopassi WA, Heitel P, Christensen KE, Cooper RI, Paton RS, Pomerantz WCK, Biggin PC, Hammond EM, Filippakopoulos P, Conway SJ.
J Med Chem (2021) 64 : 10102 -10123
PubMed 34255515 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 5 6.62 7.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5089448 1 7.00
CHEMBL5085843 1 6.80
CHEMBL5085444 1 6.50
CHEMBL3752296 1 6.50
CHEMBL5076790 1 6.30

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5089448 Kd = 100.0 nM 7.00
CHEMBL5085843 Kd = 158.49 nM 6.80
CHEMBL5085444 Kd = 316.23 nM 6.50
CHEMBL3752296 Kd = 316.23 nM 6.50
CHEMBL5076790 Kd = 501.19 nM 6.30