Assay Detail
Functional
CHEMBL5032712
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Agonist activity at human NOP receptor expressed in CHO cells assessed as stimulation of calcium mobilization by Fluo-4 AM dye based analysis
35
Total Activities
35
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Novel Mixed NOP/Opioid Receptor Peptide Agonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 34 | 7.72 | 9.29 |
| pEC50 | 1 | - | - |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL384755 | — | — | 1 | 9.29 |
| CHEMBL429363 | — | — | 1 | 9.23 |
| CHEMBL5073561 | — | — | 1 | 8.77 |
| CHEMBL5070802 | — | — | 1 | 8.70 |
| CHEMBL5093093 | — | — | 1 | 8.70 |
| CHEMBL5080536 | — | — | 1 | 8.70 |
| CHEMBL5074745 | — | — | 1 | 8.57 |
| CHEMBL5081578 | — | — | 1 | 8.55 |
| CHEMBL5079758 | — | — | 1 | 8.43 |
| CHEMBL5081993 | — | — | 1 | 8.39 |
| CHEMBL5092204 | — | — | 1 | 8.15 |
| CHEMBL5085161 | — | — | 1 | 8.03 |
| CHEMBL5086442 | — | — | 1 | 7.88 |
| CHEMBL5093399 | — | — | 1 | 7.75 |
| CHEMBL5070616 | — | — | 1 | 7.72 |
| CHEMBL5094655 | — | — | 1 | 7.58 |
| CHEMBL5094439 | — | — | 1 | 7.57 |
| CHEMBL5081139 | — | — | 1 | 7.52 |
| CHEMBL5070145 | — | — | 1 | 7.39 |
| CHEMBL5090780 | — | — | 1 | 7.31 |
| CHEMBL5072525 | — | — | 1 | 7.31 |
| CHEMBL5073730 | — | — | 1 | 7.27 |
| CHEMBL5086409 | — | — | 1 | 7.26 |
| CHEMBL5092388 | — | — | 1 | 7.25 |
| CHEMBL5072270 | — | — | 1 | 7.22 |
| CHEMBL5075880 | — | — | 1 | 7.20 |
| CHEMBL5081432 | — | — | 1 | 7.17 |
| CHEMBL5081900 | — | — | 1 | 7.07 |
| CHEMBL5079432 | — | — | 1 | 6.95 |
| CHEMBL5078005 | — | — | 1 | 6.93 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL384755 | — | EC50 | = | 0.5129 | nM | 9.29 |
| CHEMBL429363 | — | EC50 | = | 0.5888 | nM | 9.23 |
| CHEMBL5073561 | — | EC50 | = | 1.698 | nM | 8.77 |
| CHEMBL5070802 | — | EC50 | = | 1.995 | nM | 8.70 |
| CHEMBL5093093 | — | EC50 | = | 1.995 | nM | 8.70 |
| CHEMBL5080536 | — | EC50 | = | 1.995 | nM | 8.70 |
| CHEMBL5074745 | — | EC50 | = | 2.692 | nM | 8.57 |
| CHEMBL5081578 | — | EC50 | = | 2.818 | nM | 8.55 |
| CHEMBL5079758 | — | EC50 | = | 3.715 | nM | 8.43 |
| CHEMBL5081993 | — | EC50 | = | 4.074 | nM | 8.39 |
| CHEMBL5092204 | — | EC50 | = | 7.079 | nM | 8.15 |
| CHEMBL5085161 | — | EC50 | = | 9.333 | nM | 8.03 |
| CHEMBL5086442 | — | EC50 | = | 13.18 | nM | 7.88 |
| CHEMBL5093399 | — | EC50 | = | 17.78 | nM | 7.75 |
| CHEMBL5070616 | — | EC50 | = | 19.05 | nM | 7.72 |
| CHEMBL5094655 | — | EC50 | = | 26.3 | nM | 7.58 |
| CHEMBL5094439 | — | EC50 | = | 26.92 | nM | 7.57 |
| CHEMBL5081139 | — | EC50 | = | 30.2 | nM | 7.52 |
| CHEMBL5070145 | — | EC50 | = | 40.74 | nM | 7.39 |
| CHEMBL5090780 | — | EC50 | = | 48.98 | nM | 7.31 |
| CHEMBL5072525 | — | EC50 | = | 48.98 | nM | 7.31 |
| CHEMBL5073730 | — | EC50 | = | 53.7 | nM | 7.27 |
| CHEMBL5086409 | — | EC50 | = | 54.95 | nM | 7.26 |
| CHEMBL5092388 | — | EC50 | = | 56.23 | nM | 7.25 |
| CHEMBL5072270 | — | EC50 | = | 60.26 | nM | 7.22 |
| CHEMBL5075880 | — | EC50 | = | 63.1 | nM | 7.20 |
| CHEMBL5081432 | — | EC50 | = | 67.61 | nM | 7.17 |
| CHEMBL5081900 | — | EC50 | = | 85.11 | nM | 7.07 |
| CHEMBL5079432 | — | EC50 | = | 112.2 | nM | 6.95 |
| CHEMBL5078005 | — | EC50 | = | 117.49 | nM | 6.93 |
| CHEMBL5087383 | — | EC50 | = | 123.03 | nM | 6.91 |
| CHEMBL5081409 | — | EC50 | = | 151.36 | nM | 6.82 |
| CHEMBL5085090 | — | EC50 | = | 245.47 | nM | 6.61 |
| CHEMBL5091985 | — | EC50 | = | 371.54 | nM | 6.43 |
| CHEMBL285479 | — | pEC50 | - | — | - |