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Assay Detail

CHEMBL5032882

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Functional
Antiviral activity against Enterovirus D68 US/MO/14-18947 harboring 2C protein D183V/D323G drug resistant mutant by CPE assay followed by viral 2C gene sequencing
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism enterovirus D68
Confidence 1 — Organism
Curated By Autocuration

Target

enterovirus D68 (CHEMBL613204)
Type ORGANISM
Organism enterovirus D68

Publication

Discovery of Potent and Broad-Spectrum Pyrazolopyridine-Containing Antivirals against Enteroviruses D68, A71, and Coxsackievirus B3 by Targeting the Viral 2C Protein.
Hu Y, Kitamura N, Musharrafieh R, Wang J.
J Med Chem (2021) 64 : 8755 -8774
PubMed 34085827 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 5.72 5.72

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5079166 1 5.72

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5079166 EC50 = 1900.0 nM 5.72