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Assay Detail

CHEMBL5034734

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of recombinant human sEH using PHOME as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins by fluoresence-based assay
28
Total Activities
28
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Bifunctional epoxide hydrolase 2 (CHEMBL2409)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Second-Generation Dual FXR/sEH Modulators with Optimized Pharmacokinetics.
Helmstädter M, Kaiser A, Brunst S, Schmidt J, Ronchetti R, Weizel L, Proschak E, Merk D.
J Med Chem (2021) 64 : 9525 -9536
PubMed 34165993 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 28 7.64 8.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5089068 1 8.70
CHEMBL5086882 1 8.40
CHEMBL4066332 1 8.39
CHEMBL5092609 1 8.37
CHEMBL5092029 1 8.21
CHEMBL5093975 1 8.15
CHEMBL5081303 1 8.11
CHEMBL5094442 1 8.05
CHEMBL5083711 1 8.00
CHEMBL5080537 1 7.95
CHEMBL5073088 1 7.92
CHEMBL5087098 1 7.89
CHEMBL5090511 1 7.80
CHEMBL5081384 1 7.68
CHEMBL5071639 1 7.66
CHEMBL5075316 1 7.51
CHEMBL5070912 1 7.42
CHEMBL4095371 1 7.40
CHEMBL5093488 1 7.39
CHEMBL5075589 1 7.35
CHEMBL5082993 1 7.31
CHEMBL5083732 1 7.15
CHEMBL5085799 1 7.07
CHEMBL5074951 1 7.03
CHEMBL5091524 1 6.96
CHEMBL5079511 1 6.77
CHEMBL5090857 1 6.76
CHEMBL5071516 1 6.57

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5089068 IC50 = 2.0 nM 8.70
CHEMBL5086882 IC50 = 4.0 nM 8.40
CHEMBL4066332 IC50 = 4.1 nM 8.39
CHEMBL5092609 IC50 = 4.3 nM 8.37
CHEMBL5092029 IC50 = 6.1 nM 8.21
CHEMBL5093975 IC50 = 7.0 nM 8.15
CHEMBL5081303 IC50 = 7.8 nM 8.11
CHEMBL5094442 IC50 = 9.0 nM 8.05
CHEMBL5083711 IC50 = 10.0 nM 8.00
CHEMBL5080537 IC50 = 11.2 nM 7.95
CHEMBL5073088 IC50 = 12.0 nM 7.92
CHEMBL5087098 IC50 = 13.0 nM 7.89
CHEMBL5090511 IC50 = 16.0 nM 7.80
CHEMBL5081384 IC50 = 21.0 nM 7.68
CHEMBL5071639 IC50 = 22.0 nM 7.66
CHEMBL5075316 IC50 = 31.0 nM 7.51
CHEMBL5070912 IC50 = 38.0 nM 7.42
CHEMBL4095371 IC50 = 40.0 nM 7.40
CHEMBL5093488 IC50 = 41.0 nM 7.39
CHEMBL5075589 IC50 = 45.0 nM 7.35
CHEMBL5082993 IC50 = 49.0 nM 7.31
CHEMBL5083732 IC50 = 71.0 nM 7.15
CHEMBL5085799 IC50 = 85.0 nM 7.07
CHEMBL5074951 IC50 = 94.0 nM 7.03
CHEMBL5091524 IC50 = 111.0 nM 6.96
CHEMBL5079511 IC50 = 170.0 nM 6.77
CHEMBL5090857 IC50 = 175.0 nM 6.76
CHEMBL5071516 IC50 = 268.0 nM 6.57