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Assay Detail

CHEMBL5037986

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of B0AT1 (unknown origin) by radiolabled uptake assay
48
Total Activities
48
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Discovery of novel, potent and orally efficacious inhibitor of neutral amino acid transporter B<sup>0</sup>AT1 (SLC6A19).
Desai J, Patel B, Darji B, Gite A, Panchal N, Bhosale G, Shedage S, Patel S, Kadam P, Patel G, Kumar Srivastava B, Joharapurkar A, Kshirsagar S, Giri P, Bhayani H, Patel A, Ghoshdastidar K, Bandyopadhyay D, Kumar S, Jain M, Sharma R.
Bioorg Med Chem Lett (2021) 53 : 128421 -128421
PubMed 34718128 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 48 6.10 7.46

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5082788 1 7.46
CHEMBL5087496 1 7.05
CHEMBL5094524 1 7.00
CHEMBL5090717 1 6.82
CHEMBL5077170 1 6.72
CHEMBL5092865 1 6.70
CHEMBL5083821 1 6.70
CHEMBL5084448 1 6.50
CHEMBL93233 CINROMIDE 2.0 1 6.43
CHEMBL5092402 1 6.43
CHEMBL5081155 1 6.36
CHEMBL5075427 1 6.34
CHEMBL5094851 1 6.28
CHEMBL5092448 1 6.22
CHEMBL5075355 1 6.22
CHEMBL5074654 1 6.16
CHEMBL5082943 1 6.10
CHEMBL5085073 1 6.00
CHEMBL5078017 1 6.00
CHEMBL5078967 1 6.00
CHEMBL5081254 1 5.41
CHEMBL5088149 1 4.80
CHEMBL56367 NIMESULIDE 4.0 1 4.64
CHEMBL116590 1 4.15
CHEMBL5085749 1 4.11
CHEMBL5080716 1 -
CHEMBL5090681 1 -
CHEMBL5085836 1 -
CHEMBL5092903 1 -
CHEMBL5074840 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5082788 IC50 = 35.0 nM 7.46
CHEMBL5087496 IC50 = 90.0 nM 7.05
CHEMBL5094524 IC50 = 100.0 nM 7.00
CHEMBL5090717 IC50 = 150.0 nM 6.82
CHEMBL5077170 IC50 = 190.0 nM 6.72
CHEMBL5092865 IC50 = 200.0 nM 6.70
CHEMBL5083821 IC50 = 200.0 nM 6.70
CHEMBL5084448 IC50 = 320.0 nM 6.50
CHEMBL93233 CINROMIDE IC50 = 370.0 nM 6.43
CHEMBL5092402 IC50 = 370.0 nM 6.43
CHEMBL5081155 IC50 = 440.0 nM 6.36
CHEMBL5075427 IC50 = 460.0 nM 6.34
CHEMBL5094851 IC50 = 520.0 nM 6.28
CHEMBL5092448 IC50 = 600.0 nM 6.22
CHEMBL5075355 IC50 = 600.0 nM 6.22
CHEMBL5074654 IC50 = 690.0 nM 6.16
CHEMBL5082943 IC50 = 800.0 nM 6.10
CHEMBL5085073 IC50 = 1000.0 nM 6.00
CHEMBL5078017 IC50 = 1000.0 nM 6.00
CHEMBL5078967 IC50 = 1000.0 nM 6.00
CHEMBL5081254 IC50 = 3900.0 nM 5.41
CHEMBL5088149 IC50 = 16000.0 nM 4.80
CHEMBL56367 NIMESULIDE IC50 = 23000.0 nM 4.64
CHEMBL116590 IC50 = 71000.0 nM 4.15
CHEMBL5085749 IC50 = 78000.0 nM 4.11
CHEMBL5082944 IC50 > 1000.0 nM -
CHEMBL5094118 IC50 > 10000.0 nM -
CHEMBL5078865 IC50 > 1000.0 nM -
CHEMBL5074996 IC50 > 10000.0 nM -
CHEMBL5086886 IC50 > 1000.0 nM -
CHEMBL5078001 IC50 > 1000.0 nM -
CHEMBL5079561 IC50 > 1000.0 nM -
CHEMBL5086729 IC50 > 10000.0 nM -
CHEMBL5071501 IC50 > 1000.0 nM -
CHEMBL5094764 IC50 > 10000.0 nM -
CHEMBL5094598 IC50 > 10000.0 nM -
CHEMBL5077474 IC50 > 10000.0 nM -
CHEMBL5080716 IC50 > 10000.0 nM -
CHEMBL5085948 IC50 > 1000.0 nM -
CHEMBL5092919 IC50 > 10000.0 nM -
CHEMBL5083948 IC50 > 1000.0 nM -
CHEMBL5092819 IC50 > 1000.0 nM -
CHEMBL5092983 IC50 > 1000.0 nM -
CHEMBL5086307 IC50 > 10000.0 nM -
CHEMBL5074840 IC50 > 1000.0 nM -
CHEMBL5092903 IC50 > 10000.0 nM -
CHEMBL5085836 IC50 > 10000.0 nM -
CHEMBL5090681 IC50 > 10000.0 nM -