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Assay Detail

CHEMBL5039229

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against wild type Human rhinovirus B14 infected in HeLa cells assessed as reduction in virus-induced cytopathic effect incubated for 3 days by MTS/PMS assay
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism rhinovirus B14
Cell Type HeLa
Confidence 1 — Organism
Curated By Autocuration

Target

rhinovirus B14 (CHEMBL613759)
Type ORGANISM
Organism rhinovirus B14

Publication

Design, Synthesis, and Biological Evaluation of Peptidomimetic Aldehydes as Broad-Spectrum Inhibitors against Enterovirus and SARS-CoV-2.
Dai W, Jochmans D, Xie H, Yang H, Li J, Su H, Chang D, Wang J, Peng J, Zhu L, Nian Y, Hilgenfeld R, Jiang H, Chen K, Zhang L, Xu Y, Neyts J, Liu H.
J Med Chem (2022) 65 : 2794 -2808
PubMed 33872498 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 4 5.95 6.09

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5076204 1 6.09
CHEMBL5093941 1 6.01
CHEMBL477147 1 5.92
CHEMBL5085665 1 5.78

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5076204 EC50 = 810.0 nM 6.09
CHEMBL5093941 EC50 = 980.0 nM 6.01
CHEMBL477147 EC50 = 1190.0 nM 5.92
CHEMBL5085665 EC50 = 1650.0 nM 5.78