Assay Detail
Functional
CHEMBL5039834
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Antiproliferative activity against human QSG7701 cells incubated for 24 hrs by alamar blue assay
22
Total Activities
22
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | QSG7701 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Identification of a Novel TAR RNA-Binding Protein 2 Modulator with Potential Therapeutic Activity against Hepatocellular Carcinoma.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 22 | 4.21 | 4.32 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5077274 | — | — | 1 | 4.32 |
| CHEMBL5075409 | — | — | 1 | 4.30 |
| CHEMBL463499 | — | — | 1 | 4.28 |
| CHEMBL5090710 | — | — | 1 | 4.25 |
| CHEMBL5074907 | — | — | 1 | 4.25 |
| CHEMBL5084406 | — | — | 1 | 4.23 |
| CHEMBL5079841 | — | — | 1 | 4.23 |
| CHEMBL5092403 | — | — | 1 | 4.21 |
| CHEMBL5083874 | — | — | 1 | 4.21 |
| CHEMBL5088565 | — | — | 1 | 4.20 |
| CHEMBL5088504 | — | — | 1 | 4.19 |
| CHEMBL5093445 | — | — | 1 | 4.17 |
| CHEMBL5080302 | — | — | 1 | 4.17 |
| CHEMBL5084874 | — | — | 1 | 4.16 |
| CHEMBL5091460 | — | — | 1 | 4.16 |
| CHEMBL826 | ENOXACIN | 4.0 | 1 | 4.14 |
| CHEMBL5086245 | — | — | 1 | 4.13 |
| CHEMBL5089811 | — | — | 1 | 4.12 |
| CHEMBL5088112 | — | — | 1 | - |
| CHEMBL5075173 | — | — | 1 | - |
| CHEMBL5089517 | — | — | 1 | - |
| CHEMBL5089048 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5077274 | — | IC50 | = | 48350.0 | nM | 4.32 |
| CHEMBL5075409 | — | IC50 | = | 50320.0 | nM | 4.30 |
| CHEMBL463499 | — | IC50 | = | 52980.0 | nM | 4.28 |
| CHEMBL5090710 | — | IC50 | = | 56350.0 | nM | 4.25 |
| CHEMBL5074907 | — | IC50 | = | 56890.0 | nM | 4.25 |
| CHEMBL5084406 | — | IC50 | = | 59470.0 | nM | 4.23 |
| CHEMBL5079841 | — | IC50 | = | 58450.0 | nM | 4.23 |
| CHEMBL5092403 | — | IC50 | = | 61350.0 | nM | 4.21 |
| CHEMBL5083874 | — | IC50 | = | 62350.0 | nM | 4.21 |
| CHEMBL5088565 | — | IC50 | = | 63250.0 | nM | 4.20 |
| CHEMBL5088504 | — | IC50 | = | 64380.0 | nM | 4.19 |
| CHEMBL5093445 | — | IC50 | = | 67230.0 | nM | 4.17 |
| CHEMBL5080302 | — | IC50 | = | 67890.0 | nM | 4.17 |
| CHEMBL5084874 | — | IC50 | = | 69320.0 | nM | 4.16 |
| CHEMBL5091460 | — | IC50 | = | 68540.0 | nM | 4.16 |
| CHEMBL826 | ENOXACIN | IC50 | = | 72350.0 | nM | 4.14 |
| CHEMBL5086245 | — | IC50 | = | 74150.0 | nM | 4.13 |
| CHEMBL5089811 | — | IC50 | = | 75860.0 | nM | 4.12 |
| CHEMBL5088112 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5075173 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5089517 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5089048 | — | IC50 | > | 100000.0 | nM | - |