Assay Detail
Functional
CHEMBL5040271
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Anti-cancer activity against human BRCA2 complemented HR-proficient Chinese hamster VC8-B2 cells assessed as reduction in cell viability treated for 24 hrs measured 48 hrs post-recovery period by MTT assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Cricetulus griseus |
| Cell Type | VC8-B2 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Carbohydrate-Based NK1R Antagonists with Broad-Spectrum Anticancer Activity.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 4.20 | 4.20 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5083565 | — | — | 1 | 4.20 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5083565 | — | IC50 | = | 63700.0 | nM | 4.20 |