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Assay Detail

CHEMBL5040294

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against SARS-COV2 infected in HT-1080 cells expressing ACE2 preincubated for 30 mins followed by cell addition after 24 hrs by Nano-glo luciferase reagent based assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Severe acute respiratory syndrome coronavirus 2
Cell Type HT-1080
Confidence 1 — Organism
Curated By Autocuration

Target

SARS-CoV-2 (CHEMBL4303835)
Type ORGANISM
Organism Severe acute respiratory syndrome coronavirus 2

Publication

Synthetic Peptides That Antagonize the Angiotensin-Converting Enzyme-2 (ACE-2) Interaction with SARS-CoV-2 Receptor Binding Spike Protein.
Sadremomtaz A, Al-Dahmani ZM, Ruiz-Moreno AJ, Monti A, Wang C, Azad T, Bell JC, Doti N, Velasco-Velázquez MA, de Jong D, de Jonge J, Smit J, Dömling A, van Goor H, Groves MR.
J Med Chem (2022) 65 : 2836 -2847
PubMed 34328726 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.72 5.72

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5088895 1 5.72

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5088895 IC50 = 1900.0 nM 5.72