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Assay Detail

CHEMBL5041868

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of Glycosidase (unknown origin)
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

5-<i>C</i>-Branched Deoxynojirimycin: Strategy for Designing a 1-Deoxynojirimycin-Based Pharmacological Chaperone with a Nanomolar Affinity for Pompe Disease.
Kato A, Nakagome I, Kanekiyo U, Lu TT, Li YX, Yoshimura K, Kishida M, Shinzawa K, Yoshida T, Tanaka N, Jia YM, Nash RJ, Fleet GWJ, Yu CY.
J Med Chem (2022) 65 : 2329 -2341
PubMed 35072486 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 5.60 6.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5088994 1 6.70
CHEMBL5085402 1 6.10
CHEMBL5028072 1 6.00
CHEMBL5091861 1 4.92
CHEMBL5082792 1 4.30

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5088994 IC50 = 200.0 nM 6.70
CHEMBL5085402 IC50 = 800.0 nM 6.10
CHEMBL5028072 IC50 = 1000.0 nM 6.00
CHEMBL5091861 IC50 = 12000.0 nM 4.92
CHEMBL5082792 IC50 = 50000.0 nM 4.30