Assay Detail
Functional
CHEMBL5056089
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Cytotoxicity against human HT-29 cells assessed as inhibition of cell growth measured after 72 hrs by CellTiter-Glo reagent based luminescence assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HT-29 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Anticancer properties of indole derivatives as IsoCombretastatin A-4 analogues.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 9.08 | 9.08 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5082180 | — | — | 1 | 9.08 |
| CHEMBL498271 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5082180 | — | IC50 | = | 0.84 | nM | 9.08 |
| CHEMBL498271 | — | IC50 | > | 100.0 | nM | - |