Assay Detail
Binding
CHEMBL5058893
Review assay metadata, readout intent, target linkage, and publication context from the same page.
mBMMC chemotaxis
2
Total Activities
2
Compounds Tested
1
Activity Types
2
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Data for DCP probe JNJ-39758979
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.63 | 8.10 |
Assay Parameters
| Parameter | Type | Value | Units | Text |
|---|---|---|---|---|
| Assay publication | Assay publication | - | — | PMID: 14722321 |
| Target protein type | Target protein type | - | — | Mouse bone marrow mast cell (mBMMC) |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3236549 | JNJ-39758979 | 2.0 | 1 | 8.10 |
| CHEMBL5087167 | — | — | 1 | 5.16 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3236549 | JNJ-39758979 | IC50 | = | 8.0 | nM | 8.10 |
| CHEMBL5087167 | — | IC50 | = | 6900.0 | nM | 5.16 |