Assay Detail
Functional
CHEMBL5096525
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Cytotoxicity against human KMM-1 cells assessed as inhibition of cell viability incubated for 72 hrs by MTS assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | KMM-1 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Recent Update on Targeting <i>c-MYC</i> G-Quadruplexes by Small Molecules for Anticancer Therapeutics.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.10 | 5.38 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5172233 | — | — | 1 | 5.38 |
| CHEMBL1358584 | — | — | 1 | 4.81 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5172233 | — | IC50 | = | 4130.0 | nM | 5.38 |
| CHEMBL1358584 | — | IC50 | = | 15600.0 | nM | 4.81 |