Assay Detail
Binding
CHEMBL5096588
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to human InsR expressed in mouse IGF1R knockout MEF cells assessed as dissociation constant
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | MEF |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Development and Therapeutic Potential of NUAKs Inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 1 | 7.92 | 7.92 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5182271 | — | — | 1 | 7.92 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5182271 | — | Kd | = | 12.0 | nM | 7.92 |