Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL5098240

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antileishmanial activity against promastigote form of Leishmania amazonensis MHOM/BR/79/Maria assessed as inhibition of parasite growth measured after 48 hrs by resazurin staining based fluorescence analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Leishmania amazonensis
Confidence 1 — Organism
Curated By Autocuration

Target

Leishmania amazonensis (CHEMBL612877)
Type ORGANISM
Organism Leishmania amazonensis

Publication

Recent advancements in anti-leishmanial research: Synthetic strategies and structural activity relationships.
Gupta O, Pradhan T, Bhatia R, Monga V.
Eur J Med Chem (2021) 223 : 113606 -113606
PubMed 34171661 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.39 5.39

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL56234 1 5.39

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL56234 IC50 = 4110.0 nM 5.39