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Assay Detail

CHEMBL5098540

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of DENV2 His tagged NS2B (48 to 95 residues)/NS3 (1 to 185 residues) protein protein interaction
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism dengue virus type 2
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Genome polyprotein (CHEMBL5980)
Type SINGLE PROTEIN
Organism dengue virus type 2

Publication

A short survey of dengue protease inhibitor development in the past 6 years (2015-2020) with an emphasis on similarities between DENV and SARS-CoV-2 proteases.
Murtuja S, Shilkar D, Sarkar B, Sinha BN, Jayaprakash V.
Bioorg Med Chem (2021) 49 : 116415 -116415
PubMed 34601454 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 4.82 4.82

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5483017 1 4.82

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5483017 IC50 = 15000.0 nM 4.82