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Assay Detail

CHEMBL5099650

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity to wild type TTR (unknown origin) assessed as gibbs free energy change by ITC analysis
6
Total Activities
6
Compounds Tested
2
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Transthyretin (CHEMBL3194)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Development of a Highly Potent Transthyretin Amyloidogenesis Inhibitor: Design, Synthesis, and Evaluation.
Pinheiro F, Pallarès I, Peccati F, Sánchez-Morales A, Varejão N, Bezerra F, Ortega-Alarcon D, Gonzalez D, Osorio M, Navarro S, Velázquez-Campoy A, Almeida MR, Reverter D, Busqué F, Alibés R, Sodupe M, Ventura S.
J Med Chem (2022) 65 : 14673 -14691
PubMed 36306808 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
deltaG 5 - -
Kd 1 7.47 7.47

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1324 TOLCAPONE 4.0 1 7.47
CHEMBL5183147 1 -
CHEMBL5172066 1 -
CHEMBL5205412 1 -
CHEMBL5172990 1 -
CHEMBL5203058 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1324 TOLCAPONE Kd = 34.0 nM 7.47
CHEMBL5183147 deltaG = -8.9 kcal/mol -
CHEMBL5172066 deltaG = -10.3 kcal/mol -
CHEMBL5205412 deltaG = -10.2 kcal/mol -
CHEMBL5172990 deltaG = -10.4 kcal/mol -
CHEMBL5203058 deltaG = -11.2 kcal/mol -