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Assay Detail

CHEMBL5108629

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human MCF7 cells assessed as cell growth inhibition
10
Total Activities
10
Compounds Tested
2
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type MCF7
Confidence 1 — Organism
Curated By Autocuration

Target

MCF7 (CHEMBL387)
Type CELL-LINE
Organism Homo sapiens

Publication

Natural products from mangrove sediments-derived microbes: Structural diversity, bioactivities, biosynthesis, and total synthesis.
Li K, Chen S, Pang X, Cai J, Zhang X, Liu Y, Zhu Y, Zhou X.
Eur J Med Chem (2022) 230 : 114117 -114117
PubMed 35063731 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 8 6.72 6.72
GI50 2 - -

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5177929 1 6.72
CHEMBL3740584 1 6.72
CHEMBL4441305 1 6.72
CHEMBL3740707 1 6.72
CHEMBL3086649 1 6.72
CHEMBL3741748 1 6.72
CHEMBL3086650 1 6.72
CHEMBL5180764 1 -
CHEMBL467698 1 -
CHEMBL478807 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5177929 IC50 = 190.0 nM 6.72
CHEMBL3740584 IC50 = 190.0 nM 6.72
CHEMBL4441305 IC50 = 190.0 nM 6.72
CHEMBL3740707 IC50 = 190.0 nM 6.72
CHEMBL3086649 IC50 = 190.0 nM 6.72
CHEMBL3741748 IC50 = 190.0 nM 6.72
CHEMBL3086650 IC50 = 190.0 nM 6.72
CHEMBL5180764 IC50 = 7.5 ug.mL-1 -
CHEMBL467698 GI50 = 0.11 ug.mL-1 -
CHEMBL478807 GI50 = 0.11 ug.mL-1 -