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Assay Detail

CHEMBL5108752

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Nipah M1999 infected in human HeLa cells assessed as reduction in viral replication incubated for 48 to 144 hrs by reporter virus assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Henipavirus nipahense
Cell Type HeLa
Confidence 1 — Organism
Curated By Autocuration

Target

Nipah virus (CHEMBL615055)
Type ORGANISM
Organism Henipavirus nipahense

Publication

Phosphoramidate Prodrugs Continue to Deliver, The Journey of Remdesivir (GS-5734) from RSV to SARS-CoV-2.
Mackman RL.
ACS Med Chem Lett (2022) 13 : 338 -347
PubMed 35291757 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 2 6.43 7.18

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5205032 1 7.18
CHEMBL2016757 GS-441524 1.0 1 5.67

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5205032 EC50 = 66.0 nM 7.18
CHEMBL2016757 GS-441524 EC50 = 2120.0 nM 5.67