Assay Detail
Binding
CHEMBL5109340
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Inhibition of recombinant CDK2/CycE (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Current progress and novel strategies that target CDK12 for drug discovery.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.76 | 8.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL23254 | PURVALANOL B | — | 1 | 8.05 |
| CHEMBL23327 | PURVALANOLA | — | 1 | 7.46 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL23254 | PURVALANOL B | IC50 | = | 9.0 | nM | 8.05 |
| CHEMBL23327 | PURVALANOLA | IC50 | = | 35.0 | nM | 7.46 |