Assay Detail
Binding
CHEMBL5110037
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Binding affinity to 5-HT1F (unknown origin) assessed as inhibition constant
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Positron Emission Tomography (PET) Imaging Tracers for Serotonin Receptors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 8.22 | 8.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL431041 | — | — | 1 | 8.30 |
| CHEMBL105261 | — | — | 1 | 8.26 |
| CHEMBL178066 | — | — | 1 | 8.09 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL431041 | — | Ki | = | 5.0 | nM | 8.30 |
| CHEMBL105261 | — | Ki | = | 5.5 | nM | 8.26 |
| CHEMBL178066 | — | Ki | = | 8.2 | nM | 8.09 |