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Assay Detail

CHEMBL5113090

Review assay metadata, readout intent, target linkage, and publication context from the same page.

ADMET
Inhibition of CYP2C8 in human liver microsomes using amodiaquine as substrate by LC-MS/MS analysis
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Homo sapiens
Tissue Liver
Subcellular Microsome
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Cytochrome P450 2C8 (CHEMBL3721)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Discovery and Structure-Based Design of Potent Covalent PPARγ Inverse-Agonists <b>BAY-4931</b> and <b>BAY-0069</b>.
Orsi DL, Pook E, Bräuer N, Friberg A, Lienau P, Lemke CT, Stellfeld T, Brüggemeier U, Pütter V, Meyer H, Baco M, Tang S, Cherniack AD, Westlake L, Bender SA, Kocak M, Strathdee CA, Meyerson M, Eis K, Goldstein JT.
J Med Chem (2022) 65 : 14843 -14863
PubMed 36270630 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 5.27 5.37

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5187164 1 5.37
CHEMBL5207130 1 5.16

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5187164 IC50 = 4300.0 nM 5.37
CHEMBL5207130 IC50 = 7000.0 nM 5.16