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Assay Detail

CHEMBL5113740

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Functional
Antifungal activity against Candida albicans assessed as fungal growth inhibition
12
Total Activities
12
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Candida albicans
Confidence 1 — Organism
Curated By Autocuration

Target

Candida albicans (CHEMBL366)
Type ORGANISM
Organism Candida albicans

Publication

Tryptophan derived natural marine alkaloids and synthetic derivatives as promising antimicrobial agents.
Almeida MC, Resende DISP, da Costa PM, Pinto MMM, Sousa E.
Eur J Med Chem (2021) 209 : 112945 -112945
PubMed 33153766 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 12 5.17 6.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5209103 1 6.30
CHEMBL5169653 1 5.55
CHEMBL5170346 1 5.50
CHEMBL5184372 1 5.32
CHEMBL302637 NORTOPSENTIN A 1 5.17
CHEMBL292801 NORTOPSENTIN B 1 5.17
CHEMBL63208 NORTOPSENTIN C 1 5.17
CHEMBL5208629 1 5.10
CHEMBL5192861 1 4.85
CHEMBL5186502 1 4.84
CHEMBL5179552 1 4.70
CHEMBL5177565 1 4.34

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5209103 IC50 = 500.0 nM 6.30
CHEMBL5169653 IC50 = 2800.0 nM 5.55
CHEMBL5170346 IC50 = 3200.0 nM 5.50
CHEMBL5184372 IC50 = 4800.0 nM 5.32
CHEMBL302637 NORTOPSENTIN A IC50 = 6800.0 nM 5.17
CHEMBL292801 NORTOPSENTIN B IC50 = 6800.0 nM 5.17
CHEMBL63208 NORTOPSENTIN C IC50 = 6800.0 nM 5.17
CHEMBL5208629 IC50 = 7900.0 nM 5.10
CHEMBL5192861 IC50 = 14200.0 nM 4.85
CHEMBL5186502 IC50 = 14500.0 nM 4.84
CHEMBL5179552 IC50 = 19900.0 nM 4.70
CHEMBL5177565 IC50 = 45700.0 nM 4.34