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Assay Detail

CHEMBL5113741

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antifungal activity against Cryptococcus neoformans assessed as fungal growth inhibition
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Cryptococcus neoformans
Confidence 1 — Organism
Curated By Autocuration

Target

Cryptococcus neoformans (CHEMBL365)
Type ORGANISM
Organism Cryptococcus neoformans

Publication

Tryptophan derived natural marine alkaloids and synthetic derivatives as promising antimicrobial agents.
Almeida MC, Resende DISP, da Costa PM, Pinto MMM, Sousa E.
Eur J Med Chem (2021) 209 : 112945 -112945
PubMed 33153766 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 6 5.22 6.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5209103 1 6.30
CHEMBL5170346 1 5.19
CHEMBL5208629 1 5.10
CHEMBL5169653 1 4.96
CHEMBL5177565 1 4.94
CHEMBL5186502 1 4.84

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5209103 IC50 = 500.0 nM 6.30
CHEMBL5170346 IC50 = 6400.0 nM 5.19
CHEMBL5208629 IC50 = 7900.0 nM 5.10
CHEMBL5169653 IC50 = 11100.0 nM 4.96
CHEMBL5177565 IC50 = 11400.0 nM 4.94
CHEMBL5186502 IC50 = 14500.0 nM 4.84