Assay Detail
Binding
CHEMBL5114214
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to GluK5 receptor (unknown origin)
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Glutamate receptor ionotropic, kainate 5 (CHEMBL2675) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Functionalized quinoxalinones as privileged structures with broad-ranging pharmacological activities.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 4.29 | 4.58 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5193862 | — | — | 1 | 4.58 |
| CHEMBL5209119 | — | — | 1 | 4.00 |
| CHEMBL5206048 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5193862 | — | Ki | = | 26400.0 | nM | 4.58 |
| CHEMBL5209119 | — | Ki | = | 100000.0 | nM | 4.00 |
| CHEMBL5206048 | — | Ki | > | 100000.0 | nM | - |