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Assay Detail

CHEMBL5118418

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Toxicity
Cytotoxicity against human L02 cells measured after 72 hrs by MTT assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Toxicity
Organism Homo sapiens
Cell Type L02
Confidence 1 — Organism
Curated By Autocuration

Target

L02 (CHEMBL4296457)
Type CELL-LINE
Organism Homo sapiens

Publication

New brefeldin A-cinnamic acid ester derivatives as potential antitumor agents: Design, synthesis and biological evaluation.
Jiang YY, Wu S, Wu YW, Gao Y, Chong D, Sun C, Wei MY, Gu YC, Shao CL, Gu Y.
Eur J Med Chem (2022) 240 : 114598 -114598
PubMed 35849940 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 6.28 7.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL19980 BREFELDIN A 1 7.00
CHEMBL5189836 1 5.55

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL19980 BREFELDIN A IC50 = 100.0 nM 7.00
CHEMBL5189836 IC50 = 2810.0 nM 5.55