Assay Detail
Binding
CHEMBL5121304
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of xanthine oxidase (unknown origin) at 10 uM using xanthine as substrate
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Isolation and biological activity of azocine and azocane alkaloids.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.21 | 6.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1467 | ALLOPURINOL | 4.0 | 1 | 6.22 |
| CHEMBL285671 | APPARICINE | — | 1 | 6.19 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1467 | ALLOPURINOL | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL285671 | APPARICINE | IC50 | = | 650.0 | nM | 6.19 |