Assay Detail
Functional
CHEMBL5124408
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiviral activity against MHV by cell based assay
11
Total Activities
11
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Murine hepatitis virus |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Peptidomimetics: An Overview of Recent Medicinal Chemistry Efforts toward the Discovery of Novel Small Molecule Inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 11 | 6.82 | 7.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5190394 | — | — | 1 | 7.10 |
| CHEMBL5174145 | — | — | 1 | 7.10 |
| CHEMBL5184284 | — | — | 1 | 6.96 |
| CHEMBL5195656 | — | — | 1 | 6.92 |
| CHEMBL5178275 | — | — | 1 | 6.92 |
| CHEMBL5194912 | — | — | 1 | 6.89 |
| CHEMBL5188945 | — | — | 1 | 6.89 |
| CHEMBL5172701 | — | — | 1 | 6.80 |
| CHEMBL5173283 | — | — | 1 | 6.80 |
| CHEMBL5175540 | — | — | 1 | 6.70 |
| CHEMBL2315036 | — | — | 1 | 5.96 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5190394 | — | EC50 | = | 80.0 | nM | 7.10 |
| CHEMBL5174145 | — | EC50 | = | 80.0 | nM | 7.10 |
| CHEMBL5184284 | — | EC50 | = | 110.0 | nM | 6.96 |
| CHEMBL5195656 | — | EC50 | = | 120.0 | nM | 6.92 |
| CHEMBL5178275 | — | EC50 | = | 120.0 | nM | 6.92 |
| CHEMBL5194912 | — | EC50 | = | 130.0 | nM | 6.89 |
| CHEMBL5188945 | — | EC50 | = | 130.0 | nM | 6.89 |
| CHEMBL5172701 | — | EC50 | = | 160.0 | nM | 6.80 |
| CHEMBL5173283 | — | EC50 | = | 160.0 | nM | 6.80 |
| CHEMBL5175540 | — | EC50 | = | 200.0 | nM | 6.70 |
| CHEMBL2315036 | — | EC50 | = | 1100.0 | nM | 5.96 |