Assay Detail
Functional
CHEMBL5124440
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antitumor activity against human UM-SCC-38 cells assessed as cell growth inhibition
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | UM-SCC-38 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Peptidomimetics: An Overview of Recent Medicinal Chemistry Efforts toward the Discovery of Novel Small Molecule Inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 6 | 6.67 | 6.85 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4753399 | — | — | 1 | 6.85 |
| CHEMBL4749062 | — | — | 1 | 6.48 |
| CHEMBL5201949 | — | — | 1 | - |
| CHEMBL5186255 | — | — | 1 | - |
| CHEMBL5174749 | — | — | 1 | - |
| CHEMBL5173034 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4753399 | — | EC50 | = | 140.0 | nM | 6.85 |
| CHEMBL4749062 | — | EC50 | = | 330.0 | nM | 6.48 |
| CHEMBL5201949 | — | EC50 | - | — | - | |
| CHEMBL5186255 | — | EC50 | - | — | - | |
| CHEMBL5174749 | — | EC50 | - | — | - | |
| CHEMBL5173034 | — | EC50 | - | — | - |