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Assay Detail

CHEMBL5127019

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of CK1delta/epsilon (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 7 — Homologous single protein target
Curated By Autocuration

Target

Casein kinase I delta/epsilon (CHEMBL3038494)
Type PROTEIN COMPLEX
Organism Homo sapiens

Publication

Therapeutic potential of quinazoline derivatives for Alzheimer's disease: A comprehensive review.
Haghighijoo Z, Zamani L, Moosavi F, Emami S.
Eur J Med Chem (2022) 227 : 113949 -113949
PubMed 34742016 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 6.10 6.10

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3823505 1 6.10

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3823505 IC50 = 800.0 nM 6.10