Assay Detail
Functional
CHEMBL5127323
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Antagonist activity at P2Y1 receptor (unknown origin)
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Progress of thrombus formation and research on the structure-activity relationship for antithrombotic drugs.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 4 | 6.04 | 6.32 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL432028 | — | — | 1 | 6.32 |
| CHEMBL104784 | — | — | 1 | 6.08 |
| CHEMBL320924 | — | — | 1 | 5.96 |
| CHEMBL108166 | — | — | 1 | 5.80 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL432028 | — | IC50 | = | 480.0 | nM | 6.32 |
| CHEMBL104784 | — | IC50 | = | 840.0 | nM | 6.08 |
| CHEMBL320924 | — | IC50 | = | 1090.0 | nM | 5.96 |
| CHEMBL108166 | — | IC50 | = | 1600.0 | nM | 5.80 |