Assay Detail
Binding
CHEMBL5127628
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]U69593 from human KOP stably expressed in CHO cells by competitive binding assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Analgesic Opioid Ligand Discovery Based on Nonmorphinan Scaffolds Derived from Natural Sources.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 9.23 | 9.23 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2381583 | 22-THIOCYANATOSALVINORIN A | — | 1 | 9.23 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2381583 | 22-THIOCYANATOSALVINORIN A | Ki | = | 0.59 | nM | 9.23 |