Assay Detail
Binding
CHEMBL5128176
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Inhibition of HIV reverse transcriptase
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Human immunodeficiency virus |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
A score years' update in the synthesis and biological evaluation of medicinally important 2-pyridones.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 9.23 | 10.24 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL83825 | — | — | 1 | 10.24 |
| CHEMBL82439 | — | — | 1 | 8.21 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL83825 | — | IC50 | = | 0.058 | nM | 10.24 |
| CHEMBL82439 | — | IC50 | = | 6.2 | nM | 8.21 |