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Assay Detail

CHEMBL5128554

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antimalarial activity against chloroquine sensitive Plasmodium falciparum 3D7 infected in human erythrocyte assessed as inhibition of parasite growth preincubated with compound for 24 hrs followed by hypoxanthine addition and measured after 24 hrs by [3H]-hypoxanthine incorporation based liquid scintillation counter
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Plasmodium falciparum
Cell Type Erythrocyte
Confidence 1 — Organism
Curated By Autocuration

Target

Plasmodium falciparum (CHEMBL364)
Type ORGANISM
Organism Plasmodium falciparum

Publication

Spiral molecules with antimalarial activities: A review.
Yang J, Wang Y, Guan W, Su W, Li G, Zhang S, Yao H.
Eur J Med Chem (2022) 237 : 114361 -114361
PubMed 35461019 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 9.10 9.10

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2387268 1 9.10

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2387268 IC50 = 0.8 nM 9.10