Assay Detail
Binding
CHEMBL5131328
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of PARP7 (unknown origin) by HTRF assay
12
Total Activities
12
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Protein mono-ADP-ribosyltransferase TIPARP (CHEMBL2380188) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Recent Discovery of PARP7 Inhibitors as Anticancer Agents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 12 | 9.00 | 9.23 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5209116 | — | — | 1 | 9.23 |
| CHEMBL5177385 | — | — | 1 | 9.21 |
| CHEMBL5181016 | — | — | 1 | 9.19 |
| CHEMBL5190796 | — | — | 1 | 9.10 |
| CHEMBL5183629 | — | — | 1 | 9.09 |
| CHEMBL5202833 | — | — | 1 | 9.06 |
| CHEMBL5174619 | — | — | 1 | 9.02 |
| CHEMBL5173659 | — | — | 1 | 9.00 |
| CHEMBL5180425 | — | — | 1 | 8.93 |
| CHEMBL5183278 | — | — | 1 | 8.91 |
| CHEMBL5193823 | — | — | 1 | 8.69 |
| CHEMBL5204396 | — | — | 1 | 8.51 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5209116 | — | IC50 | = | 0.584 | nM | 9.23 |
| CHEMBL5177385 | — | IC50 | = | 0.6114 | nM | 9.21 |
| CHEMBL5181016 | — | IC50 | = | 0.648 | nM | 9.19 |
| CHEMBL5190796 | — | IC50 | = | 0.802 | nM | 9.10 |
| CHEMBL5183629 | — | IC50 | = | 0.806 | nM | 9.09 |
| CHEMBL5202833 | — | IC50 | = | 0.87 | nM | 9.06 |
| CHEMBL5174619 | — | IC50 | = | 0.966 | nM | 9.02 |
| CHEMBL5173659 | — | IC50 | = | 1.006 | nM | 9.00 |
| CHEMBL5180425 | — | IC50 | = | 1.173 | nM | 8.93 |
| CHEMBL5183278 | — | IC50 | = | 1.243 | nM | 8.91 |
| CHEMBL5193823 | — | IC50 | = | 2.031 | nM | 8.69 |
| CHEMBL5204396 | — | IC50 | = | 3.106 | nM | 8.51 |