Assay Detail
Binding
CHEMBL5131643
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Inhibition of JAK 1 (unknown origin)
13
Total Activities
13
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Recent Developments in the Use of Kinase Inhibitors for Management of Viral Infections.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 13 | 8.01 | 8.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3622820 | ITACITINIB | 3.0 | 1 | 8.70 |
| CHEMBL4297507 | DELGOCITINIB | 3.0 | 1 | 8.55 |
| CHEMBL1789941 | RUXOLITINIB | 4.0 | 1 | 8.48 |
| CHEMBL4238926 | — | — | 1 | 8.41 |
| CHEMBL2105759 | BARICITINIB | 4.0 | 1 | 8.23 |
| CHEMBL3301607 | FILGOTINIB | 4.0 | 1 | 8.00 |
| CHEMBL4650343 | IZENCITINIB | 2.0 | 1 | 8.00 |
| CHEMBL1078178 | MOMELOTINIB | 4.0 | 1 | 7.96 |
| CHEMBL4116008 | CERDULATINIB | 2.0 | 1 | 7.92 |
| CHEMBL4747591 | — | — | 1 | 7.77 |
| CHEMBL3655081 | ABROCITINIB | 4.0 | 1 | 7.54 |
| CHEMBL3622821 | UPADACITINIB | 4.0 | 1 | 7.37 |
| CHEMBL4577523 | GOLIDOCITINIB | 2.0 | 1 | 7.14 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3622820 | ITACITINIB | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL4297507 | DELGOCITINIB | IC50 | = | 2.8 | nM | 8.55 |
| CHEMBL1789941 | RUXOLITINIB | IC50 | = | 3.3 | nM | 8.48 |
| CHEMBL4238926 | — | IC50 | = | 3.9 | nM | 8.41 |
| CHEMBL2105759 | BARICITINIB | IC50 | = | 5.9 | nM | 8.23 |
| CHEMBL3301607 | FILGOTINIB | IC50 | = | 10.0 | nM | 8.00 |
| CHEMBL4650343 | IZENCITINIB | IC50 | = | 10.0 | nM | 8.00 |
| CHEMBL1078178 | MOMELOTINIB | IC50 | = | 11.0 | nM | 7.96 |
| CHEMBL4116008 | CERDULATINIB | IC50 | = | 12.0 | nM | 7.92 |
| CHEMBL4747591 | — | IC50 | = | 17.0 | nM | 7.77 |
| CHEMBL3655081 | ABROCITINIB | IC50 | = | 29.0 | nM | 7.54 |
| CHEMBL3622821 | UPADACITINIB | IC50 | = | 43.0 | nM | 7.37 |
| CHEMBL4577523 | GOLIDOCITINIB | IC50 | = | 73.0 | nM | 7.14 |