Assay Detail
Binding
CHEMBL5135398
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of bovine liver beta-glucosidase assessed as release of p-nitrophenol using p-nitrophenyl glycoside as substrate by spectrometric assay
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Bos taurus |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Design, synthesis and glycosidase inhibition of C-4 branched LAB and DAB derivatives.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 5 | 4.15 | 4.15 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5189075 | — | — | 1 | 4.15 |
| CHEMBL2177689 | — | — | 1 | - |
| CHEMBL5198563 | — | — | 1 | - |
| CHEMBL5192700 | — | — | 1 | - |
| CHEMBL80254 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5189075 | — | IC50 | = | 71000.0 | nM | 4.15 |
| CHEMBL2177689 | — | IC50 | = | 183000.0 | nM | - |
| CHEMBL5198563 | — | IC50 | = | 226000.0 | nM | - |
| CHEMBL5192700 | — | IC50 | = | 430000.0 | nM | - |
| CHEMBL80254 | — | IC50 | = | 638000.0 | nM | - |