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Assay Detail

CHEMBL5137622

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against SARS CoV-2 clinical isolate 2019-nCoV/USA-WA1/2020 infected in human Calu-3 cells measured after 72 hrs by plaque assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Severe acute respiratory syndrome coronavirus 2
Cell Type Calu-3
Confidence 1 — Organism
Curated By Autocuration

Target

SARS-CoV-2 (CHEMBL4303835)
Type ORGANISM
Organism Severe acute respiratory syndrome coronavirus 2

Publication

Targeting SARS-CoV-2 Proteases and Polymerase for COVID-19 Treatment: State of the Art and Future Opportunities.
Cannalire R, Cerchia C, Beccari AR, Di Leva FS, Summa V.
J Med Chem (2022) 65 : 2716 -2746
PubMed 33186044 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 7.10 7.10

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2178720 N-HYDROXYCYTIDINE -1.0 1 7.10

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2178720 N-HYDROXYCYTIDINE EC50 = 80.0 nM 7.10