Assay Detail
Functional
CHEMBL5137727
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Antiproliferative activity against human U-2OS cells assessed as cell viability
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | U2OS |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
NO-HDAC dual inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 6.02 | 6.33 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4646139 | — | — | 1 | 6.33 |
| CHEMBL4639264 | — | — | 1 | 5.71 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4646139 | — | EC50 | = | 467.74 | nM | 6.33 |
| CHEMBL4639264 | — | EC50 | = | 1949.84 | nM | 5.71 |