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Assay Detail

CHEMBL5138446

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of Trypanosoma cruzi PTR1 using folic acid as substrate in presence of NADPH by spectrophotometry
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Trypanosoma cruzi
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Examination of multiple Trypanosoma cruzi targets in a new drug discovery approach for Chagas disease.
Beltran-Hortelano I, Alcolea V, Font M, Pérez-Silanes S.
Bioorg Med Chem (2022) 58 : 116577 -116577
PubMed 35189560 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 10.42 10.42

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL34259 METHOTREXATE 4.0 1 10.42

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL34259 METHOTREXATE IC50 = 0.038 nM 10.42