Assay Detail
Binding
CHEMBL5140189
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Binding affinity to human serum albumin by fluorescence polarization assay
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Phage Display Selected Cyclic Peptide Inhibitors of Kallikrein-Related Peptidases 5 and 7 and Their <i>In Vivo</i> Delivery to the Skin.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 6 | 7.04 | 7.41 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5205331 | — | — | 1 | 7.41 |
| CHEMBL5204039 | — | — | 1 | 7.41 |
| CHEMBL5172861 | — | — | 1 | 6.93 |
| CHEMBL5203652 | — | — | 1 | 6.92 |
| CHEMBL5204199 | — | — | 1 | 6.79 |
| CHEMBL5183937 | — | — | 1 | 6.78 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5205331 | — | Kd | = | 39.0 | nM | 7.41 |
| CHEMBL5204039 | — | Kd | = | 39.0 | nM | 7.41 |
| CHEMBL5172861 | — | Kd | = | 118.0 | nM | 6.93 |
| CHEMBL5203652 | — | Kd | = | 119.0 | nM | 6.92 |
| CHEMBL5204199 | — | Kd | = | 164.0 | nM | 6.79 |
| CHEMBL5183937 | — | Kd | = | 168.0 | nM | 6.78 |