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Assay Detail

CHEMBL5140586

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of TRBP (unknown origin) - recombinant Dicer (unknown origin) protein-protein interaction incubated for 3 hrs by GST pull-down assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Discovery of a Novel Small-Molecule Inhibitor Disrupting TRBP-Dicer Interaction against Hepatocellular Carcinoma via the Modulation of microRNA Biogenesis.
Peng T, He Y, Wang T, Yu J, Ma X, Zhou Z, Sheng Y, Li L, Peng H, Li S, Zou J, Yuan Y, Zhao Y, Shi H, Li F, Liu W, Hu K, Lu X, Lu X, Zhang G, Wang F.
J Med Chem (2022) 65 : 11010 -11033
PubMed 35695407 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 4.91 4.91

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5170759 1 4.91

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5170759 IC50 = 12350.0 nM 4.91