Assay Detail
Binding
CHEMBL5140973
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to GABA A receptor (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 5 — Multiple protein complex / RNA |
| Curated By | Autocuration |
Target
GABA-A receptor; anion channel (CHEMBL2093872) ↗| Type | PROTEIN COMPLEX GROUP |
| Organism | Homo sapiens |
Publication
Therapeutic Strategies to Target the Androgen Receptor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.52 | 5.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1082407 | ENZALUTAMIDE | 4.0 | 1 | 5.52 |
| CHEMBL3183409 | APALUTAMIDE | 4.0 | 1 | 5.52 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1082407 | ENZALUTAMIDE | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL3183409 | APALUTAMIDE | IC50 | = | 3000.0 | nM | 5.52 |