Assay Detail
Functional
CHEMBL5143765
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiproliferative against in mouse Ba/F3 EGFR-Del19/T790M/C797S cells
11
Total Activities
11
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Cell Type | Ba/F3 EGFR-Del19/T790M/C797S |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Emerging Approaches to Overcome Acquired Drug Resistance Obstacles to Osimertinib in Non-Small-Cell Lung Cancer.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 11 | 7.68 | 8.45 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4443483 | — | — | 1 | 8.45 |
| CHEMBL5174418 | — | — | 1 | 8.05 |
| CHEMBL5179884 | — | — | 1 | 8.05 |
| CHEMBL5195749 | — | — | 1 | 8.00 |
| CHEMBL5195167 | — | — | 1 | 7.92 |
| CHEMBL5169450 | — | — | 1 | 7.66 |
| CHEMBL3545311 | BRIGATINIB | 4.0 | 1 | 7.17 |
| CHEMBL3353410 | OSIMERTINIB | 4.0 | 1 | 6.14 |
| CHEMBL5204787 | — | — | 1 | - |
| CHEMBL5177840 | — | — | 1 | - |
| CHEMBL5190518 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4443483 | — | IC50 | = | 3.54 | nM | 8.45 |
| CHEMBL5174418 | — | IC50 | = | 9.0 | nM | 8.05 |
| CHEMBL5179884 | — | IC50 | = | 9.0 | nM | 8.05 |
| CHEMBL5195749 | — | IC50 | = | 10.0 | nM | 8.00 |
| CHEMBL5195167 | — | IC50 | = | 12.0 | nM | 7.92 |
| CHEMBL5169450 | — | IC50 | = | 22.0 | nM | 7.66 |
| CHEMBL3545311 | BRIGATINIB | IC50 | = | 67.2 | nM | 7.17 |
| CHEMBL3353410 | OSIMERTINIB | IC50 | = | 729.6 | nM | 6.14 |
| CHEMBL5204787 | — | IC50 | <= | 100.0 | nM | - |
| CHEMBL5177840 | — | IC50 | <= | 100.0 | nM | - |
| CHEMBL5190518 | — | IC50 | <= | 100.0 | nM | - |