Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL5146832

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Rhinovirus A1B infected in human H1-HeLa cells assessed as reduction in virus induced cytopathic effect incubated for 3 days by MTT assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism rhinovirus A1B
Cell Type H1-HeLa
Confidence 1 — Organism
Curated By Autocuration

Target

rhinovirus A1B (CHEMBL613713)
Type ORGANISM
Organism rhinovirus A1B

Publication

Enteroviral replication inhibition by N-Alkyl triazolopyrimidinone derivatives through a non-capsid binding mode.
Kumar Biswas B, Soo Shin J, Malpani YR, Hwang D, Jung E, Bong Han S, Vishakantegowda AG, Jung YS.
Bioorg Med Chem Lett (2022) 64 : 128673 -128673
PubMed 35292344 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 2 6.17 6.62

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL29609 PLECONARIL 2.0 1 6.62
CHEMBL5173613 1 5.72

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL29609 PLECONARIL EC50 = 240.0 nM 6.62
CHEMBL5173613 EC50 = 1900.0 nM 5.72