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Assay Detail

CHEMBL5147364

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Induction of interferon gamma production in human Vgamma9Vdelta2 T cells pretreated with K562 cells followed by compound washout and cocultured with Vgamma9Vdelta2 T cells and measured after 60 mins by ELISA
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type Vgamma9Vdelta2 T cell
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Efficiency of bis-amidate phosphonate prodrugs.
Lentini NA, Huang X, Schladetsch MA, Hsiao CC, Wiemer DF, Wiemer AJ.
Bioorg Med Chem Lett (2022) 66 : 128724 -128724
PubMed 35405283 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 5 6.44 7.64

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5191573 1 7.64
CHEMBL4088948 1 7.52
CHEMBL4204044 1 6.64
CHEMBL5195694 1 5.24
CHEMBL5170932 1 5.14

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5191573 EC50 = 23.0 nM 7.64
CHEMBL4088948 EC50 = 30.0 nM 7.52
CHEMBL4204044 EC50 = 230.0 nM 6.64
CHEMBL5195694 EC50 = 5700.0 nM 5.24
CHEMBL5170932 EC50 = 7200.0 nM 5.14