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Assay Detail

CHEMBL5151276

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Anticancer activity against human MCF7 cells assessed as inhibition of cell growth by MTT assay
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type MCF7
Confidence 1 — Organism
Curated By Autocuration

Target

MCF7 (CHEMBL387)
Type CELL-LINE
Organism Homo sapiens

Publication

Discovery of cytotoxic natural products from Red Sea sponges: Structure and synthesis.
Khan S, Al-Fadhli AA, Tilvi S.
Eur J Med Chem (2021) 220 : 113491 -113491
PubMed 33940466 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 7 8.58 8.92

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL359744 DOXORUBICIN HYDROCHLORIDE 4.0 1 8.92
CHEMBL5188813 1 8.89
CHEMBL5196791 1 8.62
CHEMBL228073 1 8.54
CHEMBL5178910 1 8.40
CHEMBL5176424 1 8.34
CHEMBL5175638 1 8.32

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL359744 DOXORUBICIN HYDROCHLORIDE IC50 = 1.2 nM 8.92
CHEMBL5188813 IC50 = 1.3 nM 8.89
CHEMBL5196791 IC50 = 2.4 nM 8.62
CHEMBL228073 IC50 = 2.9 nM 8.54
CHEMBL5178910 IC50 = 4.0 nM 8.40
CHEMBL5176424 IC50 = 4.6 nM 8.34
CHEMBL5175638 IC50 = 4.8 nM 8.32