Assay Detail
Binding
CHEMBL5151867
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Inhibition of furin (unknown origin)
30
Total Activities
26
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Why All the Fury over Furin?
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 23 | 8.61 | 10.65 |
| IC50 | 7 | 7.39 | 9.25 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5202322 | — | — | 2 | 10.65 |
| CHEMBL5207872 | — | — | 1 | 10.65 |
| CHEMBL5207759 | — | — | 1 | 10.27 |
| CHEMBL5207183 | — | — | 1 | 9.96 |
| CHEMBL5202985 | — | — | 1 | 9.31 |
| CHEMBL5175238 | — | — | 1 | 9.30 |
| CHEMBL5184039 | — | — | 1 | 9.25 |
| CHEMBL5174341 | — | — | 1 | 9.21 |
| CHEMBL5179100 | — | — | 1 | 9.17 |
| CHEMBL5199257 | — | — | 2 | 9.10 |
| CHEMBL5207252 | — | — | 1 | 8.98 |
| CHEMBL5189192 | — | — | 1 | 8.93 |
| CHEMBL5177253 | — | — | 2 | 8.60 |
| CHEMBL3126399 | — | — | 1 | 8.42 |
| CHEMBL3126398 | — | — | 1 | 8.15 |
| CHEMBL5189148 | — | — | 1 | 7.92 |
| CHEMBL5184456 | — | — | 1 | 7.89 |
| CHEMBL5201678 | — | — | 1 | 7.78 |
| CHEMBL3126396 | — | — | 1 | 7.72 |
| CHEMBL2179435 | — | — | 1 | 7.70 |
| CHEMBL5204227 | — | — | 1 | 7.55 |
| CHEMBL3126401 | — | — | 1 | 7.34 |
| CHEMBL1808924 | — | — | 1 | 6.62 |
| CHEMBL5192439 | — | — | 1 | 5.80 |
| CHEMBL1617688 | — | — | 2 | 4.50 |
| CHEMBL5203612 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5202322 | — | Ki | = | 0.0223 | nM | 10.65 |
| CHEMBL5207872 | — | Ki | = | 0.0224 | nM | 10.65 |
| CHEMBL5207759 | — | Ki | = | 0.0538 | nM | 10.27 |
| CHEMBL5207183 | — | Ki | = | 0.11 | nM | 9.96 |
| CHEMBL5202985 | — | Ki | = | 0.491 | nM | 9.31 |
| CHEMBL5175238 | — | Ki | = | 0.504 | nM | 9.30 |
| CHEMBL5202322 | — | IC50 | = | 0.56 | nM | 9.25 |
| CHEMBL5184039 | — | IC50 | = | 0.56 | nM | 9.25 |
| CHEMBL5174341 | — | Ki | = | 0.618 | nM | 9.21 |
| CHEMBL5179100 | — | Ki | = | 0.68 | nM | 9.17 |
| CHEMBL5199257 | — | Ki | = | 0.8 | nM | 9.10 |
| CHEMBL5207252 | — | Ki | = | 1.05 | nM | 8.98 |
| CHEMBL5189192 | — | Ki | = | 1.17 | nM | 8.93 |
| CHEMBL5177253 | — | Ki | = | 2.52 | nM | 8.60 |
| CHEMBL5199257 | — | IC50 | = | 2.98 | nM | 8.53 |
| CHEMBL3126399 | — | Ki | = | 3.8 | nM | 8.42 |
| CHEMBL3126398 | — | Ki | = | 7.0 | nM | 8.15 |
| CHEMBL5177253 | — | IC50 | = | 9.53 | nM | 8.02 |
| CHEMBL5189148 | — | Ki | = | 12.0 | nM | 7.92 |
| CHEMBL5184456 | — | Ki | = | 13.0 | nM | 7.89 |
| CHEMBL5201678 | — | Ki | = | 16.7 | nM | 7.78 |
| CHEMBL3126396 | — | Ki | = | 19.0 | nM | 7.72 |
| CHEMBL2179435 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL5204227 | — | Ki | = | 28.0 | nM | 7.55 |
| CHEMBL3126401 | — | Ki | = | 46.0 | nM | 7.34 |
| CHEMBL1808924 | — | Ki | = | 238.0 | nM | 6.62 |
| CHEMBL5192439 | — | Ki | = | 1570.0 | nM | 5.80 |
| CHEMBL1617688 | — | IC50 | = | 31460.0 | nM | 4.50 |
| CHEMBL1617688 | — | IC50 | = | 33790.0 | nM | 4.47 |
| CHEMBL5203612 | — | Ki | = | 0.0088 | nM | - |