Assay Detail
Binding
CHEMBL5151874
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Inhibition of Recombinant vaccinia-expressed furin (unknown origin) using Pyr-RTKR-MCA as substrate and measured by fluorescence based assay
14
Total Activities
14
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Why All the Fury over Furin?
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 14 | 6.59 | 8.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL488769 | — | — | 1 | 8.22 |
| CHEMBL485694 | — | — | 1 | 7.92 |
| CHEMBL487946 | — | — | 1 | 7.38 |
| CHEMBL506022 | — | — | 1 | 7.34 |
| CHEMBL505581 | — | — | 1 | 7.16 |
| CHEMBL5194005 | — | — | 1 | 7.05 |
| CHEMBL205548 | — | — | 1 | 6.77 |
| CHEMBL5196320 | — | — | 1 | 6.40 |
| CHEMBL448513 | — | — | 1 | 6.39 |
| CHEMBL5209516 | — | — | 1 | 5.92 |
| CHEMBL1963286 | — | — | 1 | 5.82 |
| CHEMBL5194189 | — | — | 1 | 5.57 |
| CHEMBL5184649 | — | — | 1 | 5.26 |
| CHEMBL5191784 | — | — | 1 | 5.08 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL488769 | — | Ki | = | 6.0 | nM | 8.22 |
| CHEMBL485694 | — | Ki | = | 12.0 | nM | 7.92 |
| CHEMBL487946 | — | Ki | = | 42.0 | nM | 7.38 |
| CHEMBL506022 | — | Ki | = | 46.0 | nM | 7.34 |
| CHEMBL505581 | — | Ki | = | 69.0 | nM | 7.16 |
| CHEMBL5194005 | — | Ki | = | 89.0 | nM | 7.05 |
| CHEMBL205548 | — | Ki | = | 169.0 | nM | 6.77 |
| CHEMBL5196320 | — | Ki | = | 400.0 | nM | 6.40 |
| CHEMBL448513 | — | Ki | = | 404.0 | nM | 6.39 |
| CHEMBL5209516 | — | Ki | = | 1200.0 | nM | 5.92 |
| CHEMBL1963286 | — | Ki | = | 1500.0 | nM | 5.82 |
| CHEMBL5194189 | — | Ki | = | 2700.0 | nM | 5.57 |
| CHEMBL5184649 | — | Ki | = | 5500.0 | nM | 5.26 |
| CHEMBL5191784 | — | Ki | = | 8300.0 | nM | 5.08 |