Assay Detail
Binding
CHEMBL5152268
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Inhibition of human COX2
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
The Repertoire of Small-Molecule PET Probes for Neuroinflammation Imaging: Challenges and Opportunities beyond TSPO.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 6.03 | 6.08 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5184826 | — | — | 1 | 6.08 |
| CHEMBL5192908 | — | — | 1 | 6.00 |
| CHEMBL5206077 | — | — | 1 | 6.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5184826 | — | IC50 | = | 840.0 | nM | 6.08 |
| CHEMBL5192908 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL5206077 | — | IC50 | = | 1000.0 | nM | 6.00 |